Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50034247
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  500nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359535(CHEMBL1927163)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359535(CHEMBL1927163)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359537(CHEMBL1927167)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359540(CHEMBL1927161)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359544(CHEMBL1927168)
Affinity DataIC50:  4.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359541(CHEMBL1927162)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359536(CHEMBL1927165)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359541(CHEMBL1927162)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359542(CHEMBL1927164)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359537(CHEMBL1927167)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50357934(CHEMBL1916532)
Affinity DataIC50:  1.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359540(CHEMBL1927161)
Affinity DataIC50:  2.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359545(CHEMBL1927170)
Affinity DataIC50:  2.95E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359539(CHEMBL548279)
Affinity DataIC50:  3.98E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359543(CHEMBL1927166)
Affinity DataIC50:  6.31E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359536(CHEMBL1927165)
Affinity DataIC50:  7.94E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed