Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50041962
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419607BDBM50419607(CHEMBL1940793)
Affinity DataIC50: 4.10E+3nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419601BDBM50419601(CHEMBL1940786)
Affinity DataIC50: 6.60E+3nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419605BDBM50419605(CHEMBL1940791)
Affinity DataIC50: 8.00E+3nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419609BDBM50419609(CHEMBL1940795)
Affinity DataIC50: 8.00E+3nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50382406BDBM50382406(CHEMBL1606364)
Affinity DataIC50: 9.30E+3nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419613BDBM50419613(CHEMBL1940802)
Affinity DataIC50: 9.60E+3nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419614BDBM50419614(CHEMBL1940804)
Affinity DataIC50: 1.22E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419611BDBM50419611(CHEMBL1940797)
Affinity DataIC50: 1.24E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419608BDBM50419608(CHEMBL1940794)
Affinity DataIC50: 1.34E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419603BDBM50419603(CHEMBL1940789)
Affinity DataIC50: 1.38E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419604BDBM50419604(CHEMBL1940790)
Affinity DataIC50: 1.49E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419610BDBM50419610(CHEMBL1940796)
Affinity DataIC50: 1.71E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419606BDBM50419606(CHEMBL1940792)
Affinity DataIC50: 2.03E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419615BDBM50419615(CHEMBL1940805)
Affinity DataIC50: 2.09E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419602BDBM50419602(CHEMBL1940788)
Affinity DataIC50: 2.11E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419618BDBM50419618(CHEMBL1940803)
Affinity DataIC50: 2.38E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419612BDBM50419612(CHEMBL1940800)
Affinity DataIC50: 8.30E+4nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as inhibition of epibatidine-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419600BDBM50419600(CHEMBL1940799)
Affinity DataIC50: 1.00E+5nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as decrease in epibatidine-induced calcium mobilizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419616BDBM50419616(CHEMBL1940801)
Affinity DataIC50: 1.00E+5nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as decrease in epibatidine-induced calcium mobilizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419599BDBM50419599(CHEMBL1940798)
Affinity DataIC50: 1.00E+5nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as decrease in epibatidine-induced calcium mobilizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
The Ohio State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419617BDBM50419617(CHEMBL1940787)
Affinity DataIC50: 1.00E+5nMAssay Description:Negative allosteric modulation of human nAChR alpha4beta2 expressed in HEK ts201 cells assessed as decrease in epibatidine-induced calcium mobilizati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed