Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50034549
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364070(CHEMBL1950674)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364069(CHEMBL1950673)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364072(CHEMBL1950677)
Affinity DataEC50:  2.59E+4nMAssay Description:Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364073(CHEMBL1950672)
Affinity DataEC50:  1.93E+3nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364068(CHEMBL1950671)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50205413(CHEMBL221326 | P(1),P(4)-bis(uridin-5'-yl) tetraph...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364072(CHEMBL1950677)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364065(CHEMBL1950676)
Affinity DataEC50:  720nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364066(CHEMBL1950678)
Affinity DataEC50:  9.40E+3nMAssay Description:Agonist activity at human P2Y purinoceptor 4 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364070(CHEMBL1950674)
Affinity DataEC50:  500nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364066(CHEMBL1950678)
Affinity DataEC50:  3.61E+4nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364071(CHEMBL1950675)
Affinity DataEC50:  800nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50118239(CHEMBL130266 | UDP | Uridine diphosphate | uridine...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50118242(((2R,3S,4R,5R)-5-(6-amino-2-(methylthio)-9H-purin-...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364065(CHEMBL1950676)
Affinity DataEC50:  720nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364066(CHEMBL1950678)
Affinity DataEC50:  3.61E+4nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364072(CHEMBL1950677)
Affinity DataEC50:  2.59E+4nMAssay Description:Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50184371(CHEMBL218604 | [bis({[(2R,3S,4R,5R)-5-(6-amino-9H-...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364068(CHEMBL1950671)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364070(CHEMBL1950674)
Affinity DataEC50:  500nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364071(CHEMBL1950675)
Affinity DataEC50:  800nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364065(CHEMBL1950676)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364072(CHEMBL1950677)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364069(CHEMBL1950673)
Affinity DataEC50:  6.42E+4nMAssay Description:Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364066(CHEMBL1950678)
Affinity DataEC50:  2.46E+4nMAssay Description:Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364066(CHEMBL1950678)
Affinity DataEC50:  9.40E+3nMAssay Description:Agonist activity at human P2Y purinoceptor 4 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human P2Y purinoceptor 4 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364073(CHEMBL1950672)
Affinity DataEC50:  1.93E+3nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364070(CHEMBL1950674)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Meleagris gallopavo)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364069(CHEMBL1950673)
Affinity DataEC50:  6.90E+3nMAssay Description:Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrof...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
Bar-Ilan University

Curated by ChEMBL
LigandPNGBDBM50364069(CHEMBL1950673)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at rat P2Y purinoceptor 6 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed