Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50034276
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359842BDBM50359842(CHEMBL1928905)
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359846BDBM50359846(CHEMBL1233807)
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34038BDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359842BDBM50359842(CHEMBL1928905)
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359840BDBM50359840(CHEMBL1928903)
Affinity DataKi:  31nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359840BDBM50359840(CHEMBL1928903)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156680BDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156673BDBM50156673(2-(4,5,6,7-tetrabromo-1H-benzo[d]imidazol-2-ylthio...)
Affinity DataKi:  37nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34038BDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  43nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359841BDBM50359841(CHEMBL1928904)
Affinity DataKi:  44nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156673BDBM50156673(2-(4,5,6,7-tetrabromo-1H-benzo[d]imidazol-2-ylthio...)
Affinity DataKi:  49nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359843BDBM50359843(CHEMBL1928906)
Affinity DataKi:  55nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34055BDBM34055(iodinated benzimidazole, 21)
Affinity DataKi:  62nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359846BDBM50359846(CHEMBL1233807)
Affinity DataKi:  66nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34038BDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  71nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359841BDBM50359841(CHEMBL1928904)
Affinity DataKi:  77nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34053BDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  78nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34053BDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  80nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359846BDBM50359846(CHEMBL1233807)
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359844BDBM50359844(CHEMBL1928907)
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359846BDBM50359846(CHEMBL1233807)
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359844BDBM50359844(CHEMBL1928907)
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359841BDBM50359841(CHEMBL1928904)
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359847BDBM50359847(CHEMBL1928909)
Affinity DataKi:  93nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156670BDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  97nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359843BDBM50359843(CHEMBL1928906)
Affinity DataKi:  100nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34053BDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156673BDBM50156673(2-(4,5,6,7-tetrabromo-1H-benzo[d]imidazol-2-ylthio...)
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156680BDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  109nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34053BDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  110nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359843BDBM50359843(CHEMBL1928906)
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156670BDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359840BDBM50359840(CHEMBL1928903)
Affinity DataKi:  116nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156670BDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  133nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359843BDBM50359843(CHEMBL1928906)
Affinity DataKi:  137nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359847BDBM50359847(CHEMBL1928909)
Affinity DataKi:  139nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156670BDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)
Affinity DataKi:  139nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359842BDBM50359842(CHEMBL1928905)
Affinity DataKi:  143nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156680BDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  154nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156673BDBM50156673(2-(4,5,6,7-tetrabromo-1H-benzo[d]imidazol-2-ylthio...)
Affinity DataKi:  170nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359840BDBM50359840(CHEMBL1928903)
Affinity DataKi:  172nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359845BDBM50359845(CHEMBL1928908)
Affinity DataKi:  188nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359845BDBM50359845(CHEMBL1928908)
Affinity DataKi:  195nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359842BDBM50359842(CHEMBL1928905)
Affinity DataKi:  200nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359841BDBM50359841(CHEMBL1928904)
Affinity DataKi:  210nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156680BDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)
Affinity DataKi:  212nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34055BDBM34055(iodinated benzimidazole, 21)
Affinity DataKi:  261nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34038BDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  266nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156669BDBM50156669(4,5,6,7-tetrabromo-1H-benzimidazole | 4,5,6,7-tetr...)
Affinity DataKi:  270nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
The John Paul Ii Catholic University of Lublin

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50156669BDBM50156669(4,5,6,7-tetrabromo-1H-benzimidazole | 4,5,6,7-tetr...)
Affinity DataKi:  315nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
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