Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50034335
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  5nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360748BDBM50360748(CHEMBL1934484)
Affinity DataEC50:  6nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  8nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132472BDBM50132472((S)-2-{3-[4-(4-Fluoro-phenoxy)-benzylcarbamoyl]-4-...)
Affinity DataEC50:  13nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360747BDBM50360747(CHEMBL1934483)
Affinity DataEC50:  21nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360749BDBM50360749(CHEMBL1934485)
Affinity DataEC50:  23nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360745BDBM50360745(CHEMBL1934481)
Affinity DataEC50:  26nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360750BDBM50360750(CHEMBL1934486)
Affinity DataEC50:  37nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360746BDBM50360746(CHEMBL1934482)
Affinity DataEC50:  53nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360744BDBM50360744(CHEMBL1934480)
Affinity DataEC50:  72nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360736BDBM50360736(CHEMBL1934472)
Affinity DataEC50:  120nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Dog)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  190nMAssay Description:Agonist activity at dog PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360735BDBM50360735(CHEMBL1934471)
Affinity DataEC50:  250nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360755BDBM50360755(CHEMBL1934468)
Affinity DataEC50:  280nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360751BDBM50360751(CHEMBL1934308)
Affinity DataEC50:  470nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360751BDBM50360751(CHEMBL1934308)
Affinity DataEC50:  700nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360758BDBM50360758(CHEMBL1934313)
Affinity DataEC50:  700nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360752BDBM50360752(CHEMBL1934310)
Affinity DataEC50:  760nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360737BDBM50360737(CHEMBL1934473)
Affinity DataEC50:  810nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360754BDBM50360754(CHEMBL1934314)
Affinity DataEC50:  810nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360753BDBM50360753(CHEMBL1934312)
Affinity DataEC50:  850nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360741BDBM50360741(CHEMBL1934477)
Affinity DataEC50:  1.20E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360743BDBM50360743(CHEMBL1934479)
Affinity DataEC50:  1.50E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360739BDBM50360739(CHEMBL1934475)
Affinity DataEC50:  1.50E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360749BDBM50360749(CHEMBL1934485)
Affinity DataEC50:  1.80E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360746BDBM50360746(CHEMBL1934482)
Affinity DataEC50:  1.90E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132472BDBM50132472((S)-2-{3-[4-(4-Fluoro-phenoxy)-benzylcarbamoyl]-4-...)
Affinity DataEC50:  1.92E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360745BDBM50360745(CHEMBL1934481)
Affinity DataEC50:  2.40E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360734BDBM50360734(CHEMBL1934470)
Affinity DataEC50:  2.40E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50132472BDBM50132472((S)-2-{3-[4-(4-Fluoro-phenoxy)-benzylcarbamoyl]-4-...)
Affinity DataEC50:  2.50E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Dog)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at dog PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  3.00E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360748BDBM50360748(CHEMBL1934484)
Affinity DataEC50:  3.10E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360733BDBM50360733(CHEMBL1934469)
Affinity DataEC50:  3.40E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360742BDBM50360742(CHEMBL1934478)
Affinity DataEC50: >3.40E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360757BDBM50360757(CHEMBL1934311)
Affinity DataEC50: >3.50E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at rat PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50: >4.20E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360756BDBM50360756(CHEMBL1934309)
Affinity DataEC50:  4.40E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at mouse PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360752BDBM50360752(CHEMBL1934310)
Affinity DataEC50: >4.90E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360745BDBM50360745(CHEMBL1934481)
Affinity DataEC50: >5.20E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360751BDBM50360751(CHEMBL1934308)
Affinity DataEC50:  5.90E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360738BDBM50360738(CHEMBL1934474)
Affinity DataEC50: >6.00E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360735BDBM50360735(CHEMBL1934471)
Affinity DataEC50: >6.30E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360740BDBM50360740(CHEMBL1934476)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at mouse PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360746BDBM50360746(CHEMBL1934482)
Affinity DataEC50: >6.80E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360737BDBM50360737(CHEMBL1934473)
Affinity DataEC50: >6.80E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360737BDBM50360737(CHEMBL1934473)
Affinity DataEC50: >6.80E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50360744BDBM50360744(CHEMBL1934480)
Affinity DataEC50:  7.10E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
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