Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50034283
TargetEphrin type-A receptor 4(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359971BDBM50359971(CHEMBL1927263)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetEphrin type-A receptor 4(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359970BDBM50359970(CHEMBL1927262)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEphrin type-A receptor 4(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359969BDBM50359969(CHEMBL1927261)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed