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Found 25 Enz. Inhib. hit(s) with all data for entry = 50034293
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50335010(3-Biphenyl-4-yl-5-ethyl-4-(2-fluorophenyl)-1,2,4-t...)
Affinity DataIC50:  220nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rattus norvegicus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50335010(3-Biphenyl-4-yl-5-ethyl-4-(2-fluorophenyl)-1,2,4-t...)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]glycine from Wistar rat brain GlyT2 after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360102(CHEMBL1928735)
Affinity DataIC50:  300nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360093(CHEMBL1928737)
Affinity DataIC50:  370nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50335011(3-Biphenyl-4-yl-4-(2-fluorophenyl)-5-isopropyl-4H-...)
Affinity DataIC50:  370nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rattus norvegicus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360102(CHEMBL1928735)
Affinity DataIC50:  380nMAssay Description:Displacement of [3H]glycine from Wistar rat brain GlyT2 after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360092(CHEMBL1928736)
Affinity DataIC50:  800nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360091(CHEMBL1928738)
Affinity DataIC50:  820nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360096(CHEMBL1928741)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360094(CHEMBL1928739)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rattus norvegicus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360091(CHEMBL1928738)
Affinity DataIC50:  2.70E+3nMAssay Description:Displacement of [3H]glycine from Wistar rat brain GlyT2 after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360106(CHEMBL1928733)
Affinity DataIC50:  2.80E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360104(CHEMBL1928731)
Affinity DataIC50:  3.00E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rattus norvegicus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50335011(3-Biphenyl-4-yl-4-(2-fluorophenyl)-5-isopropyl-4H-...)
Affinity DataIC50:  3.30E+3nMAssay Description:Displacement of [3H]glycine from Wistar rat brain GlyT2 after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360095(CHEMBL1928740)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rattus norvegicus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360092(CHEMBL1928736)
Affinity DataIC50:  4.20E+3nMAssay Description:Displacement of [3H]glycine from Wistar rat brain GlyT2 after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360105(CHEMBL1928732)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360107(CHEMBL1928734)
Affinity DataIC50:  7.50E+3nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360098(CHEMBL1928743)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360097(CHEMBL1928742)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360100(CHEMBL1928745)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360101(CHEMBL1928746)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360099(CHEMBL1928744)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Rattus norvegicus)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360093(CHEMBL1928737)
Affinity DataIC50:  1.40E+4nMAssay Description:Displacement of [3H]glycine from Wistar rat brain GlyT2 after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(attus norvegicus (Rat))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50360103(CHEMBL1926706)
Affinity DataIC50:  2.20E+4nMAssay Description:Displacement of [3H]glycine from rat GlyT1 expressed in rat C6 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed