Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50034499
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50315994(CHEMBL1091604 | N-(2-((1S,2R,4R)-4-(isopropyl(meth...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363430(CHEMBL1944776)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363413(CHEMBL1946830)
Affinity DataIC50:  5.20nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363432(CHEMBL1944778)
Affinity DataIC50:  6.60nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363430(CHEMBL1944776)
Affinity DataIC50:  6.60nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363430(CHEMBL1944776)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at CCR2 by monocyte transmigration assay in pesence of 0.1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363430(CHEMBL1944776)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at CCR2 by monocyte transmigration assay in pesence of 0.5% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363415(CHEMBL1946832)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363431(CHEMBL1944777)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363423(CHEMBL1947042)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363433(CHEMBL1944779)
Affinity DataIC50:  34nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363425(CHEMBL1947044)
Affinity DataIC50:  34nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363412(CHEMBL1946829)
Affinity DataIC50:  37nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363424(CHEMBL1947043)
Affinity DataIC50:  54nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363414(CHEMBL1946831)
Affinity DataIC50:  59nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363421(CHEMBL1947040)
Affinity DataIC50:  72nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363429(CHEMBL1944780)
Affinity DataIC50:  79nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363429(CHEMBL1944780)
Affinity DataIC50:  89nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363426(CHEMBL1944773)
Affinity DataIC50:  130nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363422(CHEMBL1947041)
Affinity DataIC50:  180nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363417(CHEMBL1946834)
Affinity DataIC50:  310nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363428(CHEMBL1944775)
Affinity DataIC50:  340nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363427(CHEMBL1944774)
Affinity DataIC50:  370nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363420(CHEMBL1947039)
Affinity DataIC50:  570nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363432(CHEMBL1944778)
Affinity DataIC50:  810nMAssay Description:Displacement of [125I]MIP-1beta from CCR5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363418(CHEMBL1946835)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363416(CHEMBL1946833)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363419(CHEMBL1946836)
Affinity DataIC50:  4.10E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PMBCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50363430(CHEMBL1944776)
Affinity DataIC50:  7.30E+3nMAssay Description:Displacement of [125I]MIP-1beta from CCR5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed