Compile Data Set for Download or QSAR
maximum 50k data
Found 90 Enz. Inhib. hit(s) with all data for entry = 50034456
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362800(CHEMBL1940382)
Affinity DataKi:  8nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362810(CHEMBL1940207)
Affinity DataKi:  12.7nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362796(CHEMBL1940378)
Affinity DataKi:  14.2nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362814(CHEMBL1940203)
Affinity DataKi:  15nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362813(CHEMBL1940204)
Affinity DataKi:  20.8nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362796(CHEMBL1940378)
Affinity DataKi:  21.5nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362823(CHEMBL1940193)
Affinity DataKi:  23.9nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362803(CHEMBL1940385)
Affinity DataKi:  24.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362801(CHEMBL1940383)
Affinity DataKi:  24.8nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362802(CHEMBL1940384)
Affinity DataKi:  29.2nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362803(CHEMBL1940385)
Affinity DataKi:  29.6nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362800(CHEMBL1940382)
Affinity DataKi:  30.9nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362804(CHEMBL1940386)
Affinity DataKi:  31nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362799(CHEMBL1940381)
Affinity DataKi:  32.1nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362788(CHEMBL1940214)
Affinity DataKi:  33.7nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362795(CHEMBL1940377)
Affinity DataKi:  36.6nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362809(CHEMBL1940208)
Affinity DataKi:  40nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362812(CHEMBL1940205)
Affinity DataKi:  43nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362807(CHEMBL1940211)
Affinity DataKi:  43nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362802(CHEMBL1940384)
Affinity DataKi:  43.3nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362809(CHEMBL1940208)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362798(CHEMBL1940380)
Affinity DataKi:  47nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362810(CHEMBL1940207)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362815(CHEMBL1940202)
Affinity DataKi:  55.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362801(CHEMBL1940383)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362813(CHEMBL1940204)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362799(CHEMBL1940381)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362788(CHEMBL1940214)
Affinity DataKi:  97nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362824(CHEMBL1940192)
Affinity DataKi:  104nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362823(CHEMBL1940193)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362832(CHEMBL1940196)
Affinity DataKi:  107nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362820(CHEMBL1940197)
Affinity DataKi:  115nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362798(CHEMBL1940380)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362806(CHEMBL1940388)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362804(CHEMBL1940386)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362805(CHEMBL1940387)
Affinity DataKi:  122nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362816(CHEMBL1940201)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362795(CHEMBL1940377)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362790(CHEMBL1940216)
Affinity DataKi:  135nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362812(CHEMBL1940205)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362805(CHEMBL1940387)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362816(CHEMBL1940201)
Affinity DataKi:  144nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362797(CHEMBL1940379)
Affinity DataKi:  148nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362789(CHEMBL1940215)
Affinity DataKi:  153nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362814(CHEMBL1940203)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362806(CHEMBL1940388)
Affinity DataKi:  163nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362797(CHEMBL1940379)
Affinity DataKi:  188nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362820(CHEMBL1940197)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362831(CHEMBL1940213)
Affinity DataKi:  204nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50362808(CHEMBL1940209)
Affinity DataKi:  240nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 90 total ) | Next | Last >>
Jump to: