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Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50034572
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364441(CHEMBL1950592)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50240419((E)-1-(4-Hydroxy-3-methoxy-phenyl)-dec-4-en-3-one ...)
Affinity DataIC50:  290nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364435(CHEMBL1950598)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364436(CHEMBL1950597)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364435(CHEMBL1950598)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364440(CHEMBL1950593)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364451(CHEMBL1950584)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364445(CHEMBL1950590)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364438(CHEMBL1950595)
Affinity DataIC50:  3.60E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364448(CHEMBL1950587)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364444(CHEMBL487732)
Affinity DataIC50:  4.50E+3nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364448(CHEMBL1950587)
Affinity DataIC50:  4.80E+3nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50275147(6-Gingerol | BDBM50317427 | CHEMBL446043 | Gingero...)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364437(CHEMBL1950596)
Affinity DataIC50:  9.40E+3nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364438(CHEMBL1950595)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364439(CHEMBL1950594)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364440(CHEMBL1950593)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364449(CHEMBL1950586)
Affinity DataIC50:  1.05E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364439(CHEMBL1950594)
Affinity DataIC50:  1.11E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364447(CHEMBL1950588)
Affinity DataIC50:  1.32E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364436(CHEMBL1950597)
Affinity DataIC50:  1.43E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364446(CHEMBL1950589)
Affinity DataIC50:  1.44E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364437(CHEMBL1950596)
Affinity DataIC50:  1.58E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50240419((E)-1-(4-Hydroxy-3-methoxy-phenyl)-dec-4-en-3-one ...)
Affinity DataIC50:  1.67E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364449(CHEMBL1950586)
Affinity DataIC50:  2.26E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364443(CHEMBL1097449)
Affinity DataIC50:  3.35E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364443(CHEMBL1097449)
Affinity DataIC50:  3.51E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364442(CHEMBL1950591)
Affinity DataIC50:  3.53E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364441(CHEMBL1950592)
Affinity DataIC50:  3.82E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364442(CHEMBL1950591)
Affinity DataIC50:  3.97E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364446(CHEMBL1950589)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364445(CHEMBL1950590)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364451(CHEMBL1950584)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364450(CHEMBL1950585)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364444(CHEMBL487732)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364450(CHEMBL1950585)
Affinity DataIC50:  5.61E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364447(CHEMBL1950588)
Affinity DataIC50:  9.79E+4nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364452(CHEMBL1950583)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as inhibition of capsaicin-induced calcium influx incubated for 5 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364452(CHEMBL1950583)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50275147(6-Gingerol | BDBM50317427 | CHEMBL446043 | Gingero...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as inhibition of AITC-induced calcium influx incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364451(CHEMBL1950584)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364449(CHEMBL1950586)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364448(CHEMBL1950587)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364443(CHEMBL1097449)
Affinity DataEC50:  1.07E+4nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364442(CHEMBL1950591)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50203072(3-isothiocyanatoprop-1-ene | Allyl isothiocyanate ...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50240419((E)-1-(4-Hydroxy-3-methoxy-phenyl)-dec-4-en-3-one ...)
Affinity DataEC50:  1.60E+4nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364449(CHEMBL1950586)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50364447(CHEMBL1950588)
Affinity DataEC50:  1.43E+4nMAssay Description:Agonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50240419((E)-1-(4-Hydroxy-3-methoxy-phenyl)-dec-4-en-3-one ...)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human TRPV1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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