Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 885nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataEC50: 5.5nMAssay Description:Inverse agonist activity at histamine H3 receptor assessed as inhibition of R-alpha-methylhistamine-induced [35S]GTPgamma bindingMore data for this Ligand-Target Pair