Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50034516
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50363762(CHEMBL1947088)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]WIN35428 from human cloned DAT receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50296782((1R,2S,3S,5S)-methyl 8-((E)-3-iodoallyl)-3-p-tolyl...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]WIN35428 from human cloned DAT receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50363761(CHEMBL1947087)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]WIN35428 from human cloned DAT receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50363762(CHEMBL1947088)
Affinity DataKi:  188nMAssay Description:Displacement of [3H]nisoxetine from human cloned NET receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50363761(CHEMBL1947087)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]Citalopram from human cloned SERT receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50363761(CHEMBL1947087)
Affinity DataKi:  426nMAssay Description:Displacement of [3H]nisoxetine from human cloned NET receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50296782((1R,2S,3S,5S)-methyl 8-((E)-3-iodoallyl)-3-p-tolyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]nisoxetine from human cloned NET receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50363762(CHEMBL1947088)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]Citalopram from human cloned SERT receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed