Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50034523
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043280BDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataIC50: 0.330nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043280BDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363833BDBM50363833(CHEMBL1945010)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363826BDBM50363826(CHEMBL1947129)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363833BDBM50363833(CHEMBL1945010)
Affinity DataKd:  3.16nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363828BDBM50363828(CHEMBL1947131)
Affinity DataIC50: 4.30nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363828BDBM50363828(CHEMBL1947131)
Affinity DataKd:  4.79nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363826BDBM50363826(CHEMBL1947129)
Affinity DataKd:  6.92nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Rabbit)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82258BDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataKd:  12.6nMAssay Description:Antagonist activity at angiotensin 2 AT1 receptor in Japanese White rabbits thoracic aorta assessed as inhibition of KCl-indcuced contraction after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82258BDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 16.2nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363829BDBM50363829(CHEMBL1945006)
Affinity DataIC50: 30.6nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363830BDBM50363830(CHEMBL1945007)
Affinity DataIC50: 30.8nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363825BDBM50363825(CHEMBL1947128)
Affinity DataIC50: 52.5nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363832BDBM50363832(CHEMBL1945009)
Affinity DataIC50: 57.6nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363834BDBM50363834(CHEMBL1945148)
Affinity DataIC50: 106nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363835BDBM50363835(CHEMBL1945149)
Affinity DataIC50: 198nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363831BDBM50363831(CHEMBL1945008)
Affinity DataIC50: 214nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363827BDBM50363827(CHEMBL1947130)
Affinity DataIC50: 326nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT1 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363826BDBM50363826(CHEMBL1947129)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363832BDBM50363832(CHEMBL1945009)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363835BDBM50363835(CHEMBL1945149)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363833BDBM50363833(CHEMBL1945010)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363831BDBM50363831(CHEMBL1945008)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363828BDBM50363828(CHEMBL1947131)
Affinity DataIC50: 3.60E+3nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82258BDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363830BDBM50363830(CHEMBL1945007)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363827BDBM50363827(CHEMBL1947130)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Beijing Institute of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363829BDBM50363829(CHEMBL1945006)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]Sar1 Ile8-Ang 2 from angiotensin 2 AT2 receptor after 180 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed