Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50034659
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365814BDBM50365814(CHEMBL1956993)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365815BDBM50365815(CHEMBL1956994)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365831BDBM50365831(CHEMBL1957010)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365822BDBM50365822(CHEMBL1957001)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365809BDBM50365809(CHEMBL1956990)
Affinity DataKi:  0.160nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365812BDBM50365812(CHEMBL1956991)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365820BDBM50365820(CHEMBL1956999)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365828BDBM50365828(CHEMBL1957007)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365830BDBM50365830(CHEMBL1957009)
Affinity DataKi:  0.270nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365821BDBM50365821(CHEMBL1957000)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365818BDBM50365818(CHEMBL1956997)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365824BDBM50365824(CHEMBL1957003)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365826BDBM50365826(CHEMBL1957005)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365813BDBM50365813(CHEMBL1956992)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365827BDBM50365827(CHEMBL1957006)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365810BDBM50365810(CHEMBL1956987)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365829BDBM50365829(CHEMBL1957008)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365811BDBM50365811(CHEMBL1956988)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365817BDBM50365817(CHEMBL1956996)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365825BDBM50365825(CHEMBL1957004)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365816BDBM50365816(CHEMBL1956995)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365819BDBM50365819(CHEMBL1956998)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50222869BDBM50222869(6-(4-fluorophenoxy)-3-{[(3S)-1-isopropylpiperidin-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365832BDBM50365832(CHEMBL1957011)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365823BDBM50365823(CHEMBL1957002)
Affinity DataKi:  6.60nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Prosidion

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50365808BDBM50365808(CHEMBL1956989)
Affinity DataKi:  6.70nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365820BDBM50365820(CHEMBL1956999)
Affinity DataIC50: 129nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365817BDBM50365817(CHEMBL1956996)
Affinity DataIC50: 130nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365812BDBM50365812(CHEMBL1956991)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365819BDBM50365819(CHEMBL1956998)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365809BDBM50365809(CHEMBL1956990)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222869BDBM50222869(6-(4-fluorophenoxy)-3-{[(3S)-1-isopropylpiperidin-...)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365822BDBM50365822(CHEMBL1957001)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365808BDBM50365808(CHEMBL1956989)
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365811BDBM50365811(CHEMBL1956988)
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365823BDBM50365823(CHEMBL1957002)
Affinity DataIC50: 9.55E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365816BDBM50365816(CHEMBL1956995)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365813BDBM50365813(CHEMBL1956992)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365825BDBM50365825(CHEMBL1957004)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365833BDBM50365833(CHEMBL1957012)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365826BDBM50365826(CHEMBL1957005)
Affinity DataIC50: 3.31E+4nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50365829BDBM50365829(CHEMBL1957008)
Affinity DataIC50: 3.31E+4nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed