Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50039537
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379660(CHEMBL2013185)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379656(CHEMBL2013181)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50356121(CHEMBL1962712 | CHEMBL1909781)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379662(CHEMBL2013186)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379659(CHEMBL2013184)
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379655(CHEMBL2013178)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379657(CHEMBL2013182)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379660(CHEMBL2013185)
Affinity DataIC50: 1.90E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379656(CHEMBL2013181)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379655(CHEMBL2013178)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379658(CHEMBL2013183)
Affinity DataIC50: 2.12E+5nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379663(CHEMBL2013179)
Affinity DataIC50: 2.31E+5nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379657(CHEMBL2013182)
Affinity DataIC50: 2.37E+5nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379658(CHEMBL2013183)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50356121(CHEMBL1962712 | CHEMBL1909781)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379657(CHEMBL2013182)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379658(CHEMBL2013183)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379662(CHEMBL2013186)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50356121(CHEMBL1962712 | CHEMBL1909781)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379663(CHEMBL2013179)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379655(CHEMBL2013178)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379656(CHEMBL2013181)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379660(CHEMBL2013185)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379659(CHEMBL2013184)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379663(CHEMBL2013179)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379654(CHEMBL2013180)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379659(CHEMBL2013184)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of tPA using CH3SO2-D-HHT-Gly-Arg-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379654(CHEMBL2013180)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379662(CHEMBL2013186)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of plasmin using tosyl-Gly-Pro-Lys-pNA as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Louisville

Curated by ChEMBL
LigandPNGBDBM50379654(CHEMBL2013180)
Affinity DataIC50: 2.79E+5nMAssay Description:Inhibition of urokinase-type plasminogen activator using Glt-Gly-Arg-AMC as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed