Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50034687
TargetSphingosine 1-phosphate receptor 1(Rat)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at rat S1P1 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataEC50:  0.370nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363937(CHEMBL1951588)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364607(CHEMBL1951304)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at rat S1P1 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Rat)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363937(CHEMBL1951588)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at rat S1P1 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSphingosine 1-phosphate receptor 1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364607(CHEMBL1951304)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human S1P1 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364607(CHEMBL1951304)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human S1P5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364607(CHEMBL1951304)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human S1P4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50363937(CHEMBL1951588)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50364607(CHEMBL1951304)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor expressed in CHO-K1 cells assessed as induction of GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed