Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50039569
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380131BDBM50380131(CHEMBL2013231)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human CXCR7 expressed in HEK293T cells co-expressing beta-arrestin2-YFP assessed as beta-arrestin2 recruitment after 1 hr by BRET...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380130BDBM50380130(CHEMBL2013230)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human CXCR7 expressed in HEK293T cells co-expressing beta-arrestin2-YFP assessed as beta-arrestin2 recruitment after 1 hr by BRET...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380130BDBM50380130(CHEMBL2013230)
Affinity DataKi:  7.94nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380114BDBM50380114(CHEMBL2013216)
Affinity DataKi:  12.6nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380130BDBM50380130(CHEMBL2013230)
Affinity DataEC50:  14.1nMAssay Description:Agonist activity at human CXCR7 expressed in HEK293 cells assessed as reduction of receptor surface expression after 1 hr by ELISA based internalizat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380134BDBM50380134(CHEMBL2013215)
Affinity DataKi:  15.8nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380131BDBM50380131(CHEMBL2013231)
Affinity DataKi:  19.9nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380131BDBM50380131(CHEMBL2013231)
Affinity DataEC50:  23.7nMAssay Description:Agonist activity at human CXCR7 expressed in HEK293 cells assessed as reduction of receptor surface expression after 1 hr by ELISA based internalizat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380121BDBM50380121(CHEMBL2013219)
Affinity DataKi:  25.1nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380123BDBM50380123(CHEMBL2013222)
Affinity DataKi:  31.6nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380125BDBM50380125(CHEMBL2013224)
Affinity DataKi:  50.1nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380126BDBM50380126(CHEMBL2013225)
Affinity DataKi:  79.4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380136BDBM50380136(CHEMBL2013226)
Affinity DataKi:  79.4nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380124BDBM50380124(CHEMBL2013223)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380127BDBM50380127(CHEMBL2013227)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380118BDBM50380118(CHEMBL2013214)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380116BDBM50380116(CHEMBL2013212)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380119BDBM50380119(CHEMBL2013217)
Affinity DataKi:  794nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380122BDBM50380122(CHEMBL2013220)
Affinity DataKi:  794nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380135BDBM50380135(CHEMBL2013221)
Affinity DataKi:  794nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380132BDBM50380132(CHEMBL2010828)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380120BDBM50380120(CHEMBL2013218)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380137BDBM50380137(CHEMBL2013232)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380128BDBM50380128(CHEMBL2013228)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human CXCR7 expressed in HEK293T cells co-expressing beta-arrestin2-YFP assessed as beta-arrestin2 recruitment after 1 hr by BRET...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380115BDBM50380115(CHEMBL2013233)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380117BDBM50380117(CHEMBL2013213)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380133BDBM50380133(CHEMBL2013234)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380128BDBM50380128(CHEMBL2013228)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380129BDBM50380129(CHEMBL2013229)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed