Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50039947
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Bmssi Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386735BDBM50386735(CHEMBL404782)
Affinity DataIC50: 170nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux expressed in HEK293 cells after 48 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Bmssi Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386736BDBM50386736(CHEMBL406837)
Affinity DataIC50: 260nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux expressed in HEK293 cells after 48 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Bmssi Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386738BDBM50386738(CHEMBL1834565)
Affinity DataIC50: 270nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux expressed in HEK293 cells after 48 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Bmssi Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386734BDBM50386734(CHEMBL260654)
Affinity DataIC50: 350nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux expressed in HEK293 cells after 48 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Bmssi Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386739BDBM50386739(CHEMBL1834568)
Affinity DataIC50: 350nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux expressed in HEK293 cells after 48 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Bmssi Umr 5086 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386737BDBM50386737(CHEMBL1834566)
Affinity DataIC50: 450nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux expressed in HEK293 cells after 48 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed