Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50004628
TargetIntegrase(Human immunodeficiency virus type 1)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50484988(CHEMBL2018722)
Affinity DataIC50: 3.84E+4nMAssay Description:Inhibition of GST-tagged HIV1 integrase and C-terminal His6-tagged HIV1 integrase dimerization after 3 hrs by AlphaScreen-based dimerization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50484988(CHEMBL2018722)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of HIV1 integrase using oligodeoxynucleotide as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50484987(CHEMBL2018721)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of GST-tagged HIV1 integrase and C-terminal His6-tagged HIV1 integrase dimerization after 3 hrs by AlphaScreen-based dimerization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed