Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50039662
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381886BDBM50381886(CHEMBL2022363)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381882BDBM50381882(CHEMBL2022694)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50180036BDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  1.82nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381885BDBM50381885(CHEMBL2022364)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381883BDBM50381883(CHEMBL2022692)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381888BDBM50381888(CHEMBL2022361)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200170BDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  4.35nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381880BDBM50381880(CHEMBL2022698)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381887BDBM50381887(CHEMBL2022362)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381886BDBM50381886(CHEMBL2022363)
Affinity DataKi:  11.6nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381889BDBM50381889(CHEMBL2022360)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381888BDBM50381888(CHEMBL2022361)
Affinity DataKi:  16.5nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381873BDBM50381873(CHEMBL2022696)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381875BDBM50381875(CHEMBL2022703)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381880BDBM50381880(CHEMBL2022698)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381883BDBM50381883(CHEMBL2022692)
Affinity DataKi:  64.6nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381889BDBM50381889(CHEMBL2022360)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381873BDBM50381873(CHEMBL2022696)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381884BDBM50381884(CHEMBL2022365)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381875BDBM50381875(CHEMBL2022703)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50180036BDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200170BDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381878BDBM50381878(CHEMBL2022700)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381881BDBM50381881(CHEMBL2022695)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381885BDBM50381885(CHEMBL2022364)
Affinity DataKi:  206nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381882BDBM50381882(CHEMBL2022694)
Affinity DataKi:  234nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381876BDBM50381876(CHEMBL2022702)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381887BDBM50381887(CHEMBL2022362)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381884BDBM50381884(CHEMBL2022365)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381879BDBM50381879(CHEMBL2022699)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381881BDBM50381881(CHEMBL2022695)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381877BDBM50381877(CHEMBL2022701)
Affinity DataKi:  916nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381879BDBM50381879(CHEMBL2022699)
Affinity DataKi:  950nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381878BDBM50381878(CHEMBL2022700)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381876BDBM50381876(CHEMBL2022702)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381874BDBM50381874(CHEMBL2022697)
Affinity DataKi:  7.90E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381874BDBM50381874(CHEMBL2022697)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381877BDBM50381877(CHEMBL2022701)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed