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Report error Found 135 Enz. Inhib. hit(s) with all data for entry = 50039840
Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50151982(5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50151982(5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384954(CHEMBL2037521)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


Target5-hydroxytryptamine receptor 2A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384965(CHEMBL2037529)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384966(CHEMBL2037530)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384969(CHEMBL2037431)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384955(CHEMBL2037522)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363900(CHEMBL1946258)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384954(CHEMBL2037521)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384962(CHEMBL2037526)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384954(CHEMBL2037521)
Affinity DataKi:  26.5nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384964(CHEMBL2037528)
Affinity DataKi:  28.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363897(CHEMBL1946254)
Affinity DataKi:  28.6nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384955(CHEMBL2037522)
Affinity DataKi:  30.8nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384968(CHEMBL2037430)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363898(CHEMBL1946255)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384955(CHEMBL2037522)
Affinity DataKi:  35.6nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384968(CHEMBL2037430)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384959(CHEMBL2037518)
Affinity DataKi:  44.4nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistamine H1 receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384964(CHEMBL2037528)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]Pyrilamine from human H1 histamine receptor by liquid scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent noradrenaline transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]Nisoxetine from human NET by liquid scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384960(CHEMBL2037519)
Affinity DataKi:  51.5nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHistamine H1 receptor(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]Pyrilamine from human H1 histamine receptor by liquid scintillation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384966(CHEMBL2037530)
Affinity DataKi:  62.6nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384960(CHEMBL2037519)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363899(CHEMBL1946257)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363897(CHEMBL1946254)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384955(CHEMBL2037522)
Affinity DataKi:  65.5nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataKi:  72nMAssay Description:Binding affinity to human 5HT2C receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384964(CHEMBL2037528)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384959(CHEMBL2037518)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384969(CHEMBL2037431)
Affinity DataKi:  90.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384964(CHEMBL2037528)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384962(CHEMBL2037526)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384966(CHEMBL2037530)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384956(CHEMBL2037523)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363900(CHEMBL1946258)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384961(CHEMBL2037520)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384969(CHEMBL2037431)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384970(CHEMBL2037432)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384956(CHEMBL2037523)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50363897(CHEMBL1946254)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384962(CHEMBL2037526)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSodium-dependent serotonin transporter(Human)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384969(CHEMBL2037431)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]Citalopram from human SERT by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50384967(CHEMBL2037531)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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