Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50039765
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383675BDBM50383675(CHEMBL2030074)
Affinity DataEC50:  77nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383674BDBM50383674(CHEMBL2030073)
Affinity DataEC50:  97nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383678BDBM50383678(CHEMBL2030077)
Affinity DataEC50:  120nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383673BDBM50383673(CHEMBL2030072)
Affinity DataEC50:  120nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383676BDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383682BDBM50383682(CHEMBL2030081)
Affinity DataEC50:  330nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383684BDBM50383684(CHEMBL1961795)
Affinity DataEC50:  400nMAssay Description:Agonist activity at Rev-erbalpha assessed as NCoR recruitment by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383677BDBM50383677(CHEMBL2030076)
Affinity DataEC50:  600nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383680BDBM50383680(CHEMBL2030079)
Affinity DataEC50:  620nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383661BDBM50383661(CHEMBL2030064)
Affinity DataEC50:  650nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383672BDBM50383672(CHEMBL2030071)
Affinity DataEC50:  650nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383683BDBM50383683(CHEMBL2030082)
Affinity DataEC50:  710nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383681BDBM50383681(CHEMBL2030080)
Affinity DataEC50:  780nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383671BDBM50383671(CHEMBL2030070)
Affinity DataEC50:  800nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383668BDBM50383668(CHEMBL2029898)
Affinity DataEC50:  840nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383666BDBM50383666(CHEMBL2029886)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383669BDBM50383669(CHEMBL2030065)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383665BDBM50383665(CHEMBL2029885)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383679BDBM50383679(CHEMBL2030078)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383664BDBM50383664(CHEMBL2029883)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383684BDBM50383684(CHEMBL1961795)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383663BDBM50383663(CHEMBL2029882)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383662BDBM50383662(CHEMBL2029876)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383667BDBM50383667(CHEMBL2029895)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50383670BDBM50383670(CHEMBL2030069)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed