Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50040856
TargetOxysterols receptor LXR-beta(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human LXR-beta assessed as increase in recruitment of Trap 220/D22 coactivator peptide by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | [3H]T0901317 | T 0901317 | N-[4-(1,1...)
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity at human LXR-alpha assessed as increase in recruitment of Trap 220/Drip2 coactivator peptide by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50401084(CHEMBL2204435)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human LXR-alpha assessed as increase in recruitment of Trap 220/Drip2 coactivator peptide by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50401084(CHEMBL2204435)
Affinity DataEC50:  3.04E+3nMAssay Description:Agonist activity at human LXR-beta assessed as increase in recruitment of Trap 220/D22 coactivator peptide by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50401084(CHEMBL2204435)
Affinity DataEC50:  3.78E+4nMAssay Description:Transactivation of human LXR-beta transfected in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50401084(CHEMBL2204435)
Affinity DataEC50:  8.08E+4nMAssay Description:Transactivation of human LXR-alpha transfected in HEK293 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed