Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50039799
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384358BDBM50384358(CHEMBL2031027 | US9346795, 92)
Affinity DataIC50: 9nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384358BDBM50384358(CHEMBL2031027 | US9346795, 92)
Affinity DataIC50: 10nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384355BDBM50384355(CHEMBL2031024 | US9346795, 91)
Affinity DataIC50: 12nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384341BDBM50384341(CHEMBL2031029)
Affinity DataIC50: 14nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384347BDBM50384347(CHEMBL2031016)
Affinity DataIC50: 15nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384353BDBM50384353(CHEMBL2031022 | US9346795, 59)
Affinity DataIC50: 16nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384341BDBM50384341(CHEMBL2031029)
Affinity DataIC50: 16nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384347BDBM50384347(CHEMBL2031016)
Affinity DataIC50: 17nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384352BDBM50384352(CHEMBL2031021 | US9346795, 53)
Affinity DataIC50: 17nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384360BDBM50384360(CHEMBL2031030)
Affinity DataIC50: 19nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384359BDBM50384359(CHEMBL2031028)
Affinity DataIC50: 22nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384356BDBM50384356(CHEMBL2031025 | US9346795, 105)
Affinity DataIC50: 22nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384350BDBM50384350(CHEMBL2031019)
Affinity DataIC50: 23nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384344BDBM50384344(CHEMBL2031012 | US9346795, 1)
Affinity DataIC50: 24nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384362BDBM50384362(CHEMBL2031032)
Affinity DataIC50: 26nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384362BDBM50384362(CHEMBL2031032)
Affinity DataIC50: 26nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384356BDBM50384356(CHEMBL2031025 | US9346795, 105)
Affinity DataIC50: 29nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384350BDBM50384350(CHEMBL2031019)
Affinity DataIC50: 32nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384344BDBM50384344(CHEMBL2031012 | US9346795, 1)
Affinity DataIC50: 32nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384348BDBM50384348(CHEMBL2031017 | US9346795, 7)
Affinity DataIC50: 35nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384355BDBM50384355(CHEMBL2031024 | US9346795, 91)
Affinity DataIC50: 35nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384342BDBM50384342(CHEMBL2031010)
Affinity DataIC50: 35nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384349BDBM50384349(CHEMBL2031018 | US9346795, 11)
Affinity DataIC50: 37nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384348BDBM50384348(CHEMBL2031017 | US9346795, 7)
Affinity DataIC50: 37nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384357BDBM50384357(CHEMBL2031026 | US9346795, 116)
Affinity DataIC50: 37nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384363BDBM50384363(CHEMBL2031014 | US9346795, 27)
Affinity DataIC50: 41nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384353BDBM50384353(CHEMBL2031022 | US9346795, 59)
Affinity DataIC50: 44nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384357BDBM50384357(CHEMBL2031026 | US9346795, 116)
Affinity DataIC50: 47nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384349BDBM50384349(CHEMBL2031018 | US9346795, 11)
Affinity DataIC50: 47nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384360BDBM50384360(CHEMBL2031030)
Affinity DataIC50: 47nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384346BDBM50384346(CHEMBL2031015)
Affinity DataIC50: 54nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384361BDBM50384361(CHEMBL2031031 | US9346795, 96)
Affinity DataIC50: 62nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384352BDBM50384352(CHEMBL2031021 | US9346795, 53)
Affinity DataIC50: 78nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384363BDBM50384363(CHEMBL2031014 | US9346795, 27)
Affinity DataIC50: 110nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384361BDBM50384361(CHEMBL2031031 | US9346795, 96)
Affinity DataIC50: 120nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384359BDBM50384359(CHEMBL2031028)
Affinity DataIC50: 140nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384345BDBM50384345(CHEMBL2031013)
Affinity DataIC50: 150nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384345BDBM50384345(CHEMBL2031013)
Affinity DataIC50: 180nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384351BDBM50384351(CHEMBL2031020)
Affinity DataIC50: 280nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384346BDBM50384346(CHEMBL2031015)
Affinity DataIC50: 400nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384351BDBM50384351(CHEMBL2031020)
Affinity DataIC50: 550nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384354BDBM50384354(CHEMBL2031023)
Affinity DataIC50: 590nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384354BDBM50384354(CHEMBL2031023)
Affinity DataIC50: 710nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetApoptosis regulator Bcl-2(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384343BDBM50384343(CHEMBL2031011)
Affinity DataIC50: 910nMAssay Description:Inhibition in GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384343BDBM50384343(CHEMBL2031011)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Bristol-Myers Squibb Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384342BDBM50384342(CHEMBL2031010)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Bcl-XL using fluoresceinated 18-mer Bim as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed