Found 23 Enz. Inhib. hit(s) with all data for entry = 50039801 
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cephalon
Curated by ChEMBL
Cephalon
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Inverse agonist activity at human H3 receptor by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
