Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50039802
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384423BDBM50384423(CHEMBL2031485 | US9896452, Example 62)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384412BDBM50384412(CHEMBL2031504)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384437BDBM50384437(CHEMBL2031501)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384436BDBM50384436(CHEMBL2031500)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384408BDBM50384408(CHEMBL2031498)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384429BDBM50384429(CHEMBL2031492 | US9896452, Example 137)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384428BDBM50384428(CHEMBL2031491 | US9896452, Example 8)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384417BDBM50384417(CHEMBL2031478)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384408BDBM50384408(CHEMBL2031498)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384417BDBM50384417(CHEMBL2031478)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384419BDBM50384419(CHEMBL2031480)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384419BDBM50384419(CHEMBL2031480)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384418BDBM50384418(CHEMBL2031479)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384430BDBM50384430(CHEMBL2031493 | US9896452, Example 12)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384420BDBM50384420(CHEMBL2031482)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384415BDBM50384415(CHEMBL2031507)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384411BDBM50384411(CHEMBL2031503)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384411BDBM50384411(CHEMBL2031503)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384426BDBM50384426(CHEMBL2031489 | US9896452, Example 9)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384420BDBM50384420(CHEMBL2031482)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384421BDBM50384421(CHEMBL2031483)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384422BDBM50384422(CHEMBL2031484 | US9896452, Example 125)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384412BDBM50384412(CHEMBL2031504)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384423BDBM50384423(CHEMBL2031485 | US9896452, Example 62)
Affinity DataIC50: 8.70nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384409BDBM50384409(CHEMBL2031487 | US9896452, Example 138)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384427BDBM50384427(CHEMBL2031490 | US9896452, Example 139)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384413BDBM50384413(CHEMBL2031505)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384436BDBM50384436(CHEMBL2031500)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384421BDBM50384421(CHEMBL2031483)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384414BDBM50384414(CHEMBL2031506)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384424BDBM50384424(CHEMBL2031486 | US9896452, Example 124)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384418BDBM50384418(CHEMBL2031479)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384435BDBM50384435(CHEMBL2031499)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384416BDBM50384416(CHEMBL291536 | CHEMBL2111553 | SB-334867)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384431BDBM50384431(CHEMBL2031494)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384427BDBM50384427(CHEMBL2031490 | US9896452, Example 139)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384409BDBM50384409(CHEMBL2031487 | US9896452, Example 138)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384426BDBM50384426(CHEMBL2031489 | US9896452, Example 9)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384428BDBM50384428(CHEMBL2031491 | US9896452, Example 8)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384431BDBM50384431(CHEMBL2031494)
Affinity DataIC50: 62nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384429BDBM50384429(CHEMBL2031492 | US9896452, Example 137)
Affinity DataIC50: 82nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384414BDBM50384414(CHEMBL2031506)
Affinity DataIC50: 96nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384410BDBM50384410(CHEMBL2031502)
Affinity DataIC50: 121nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384415BDBM50384415(CHEMBL2031507)
Affinity DataIC50: 125nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384435BDBM50384435(CHEMBL2031499)
Affinity DataIC50: 137nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384425BDBM50384425(CHEMBL2031488)
Affinity DataIC50: 145nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384432BDBM50384432(CHEMBL2031495)
Affinity DataIC50: 146nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384413BDBM50384413(CHEMBL2031505)
Affinity DataIC50: 151nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384424BDBM50384424(CHEMBL2031486 | US9896452, Example 124)
Affinity DataIC50: 221nMAssay Description:Antagonist activity at OX2 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Scripps Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50384434BDBM50384434(CHEMBL2031497)
Affinity DataIC50: 390nMAssay Description:Antagonist activity at OX1 receptor expressed in CHO cells assessed as inhibition of OXA-stimulated intracellular calcium mobilization after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
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