Compile Data Set for Download or QSAR
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Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 50040493
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50049479((S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-a...)
Affinity DataIC50:  6.08nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  15.9nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394979(CHEMBL18872)
Affinity DataIC50:  62.9nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395006(CHEMBL2163473)
Affinity DataIC50:  465nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))
Affinity DataIC50:  568nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394997(CHEMBL2163482 | US9708370, DBG-253-6)
Affinity DataIC50:  723nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395005(CHEMBL2163474)
Affinity DataIC50:  729nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395009(CHEMBL2163470)
Affinity DataIC50:  750nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394996(CHEMBL2163348 | US9708370, DBG-253-7)
Affinity DataIC50:  771nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)
Affinity DataIC50:  808nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395009(CHEMBL2163470)
Affinity DataIC50:  1.11E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394983(CHEMBL2163466)
Affinity DataIC50:  1.17E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataIC50:  1.34E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394999(CHEMBL2163480 | US9708370, DBG-253-3)
Affinity DataIC50:  1.34E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395004(CHEMBL2163475)
Affinity DataIC50:  1.64E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395007(CHEMBL2163472)
Affinity DataIC50:  1.80E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50049479((S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-a...)
Affinity DataIC50:  1.82E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  2.08E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataIC50:  2.77E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataIC50:  2.89E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394995(CHEMBL2163483 | US9708370, DBG-253-8)
Affinity DataIC50:  3.25E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394985(CHEMBL2163464)
Affinity DataIC50:  3.61E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394998(CHEMBL2163481 | US9708370, DBG-253-5)
Affinity DataIC50:  3.74E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394986(CHEMBL2163463)
Affinity DataIC50:  3.86E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394982(CHEMBL2163467)
Affinity DataIC50:  4.55E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394984(CHEMBL2163465)
Affinity DataIC50:  5.41E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))
Affinity DataIC50:  6.06E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395019(CHEMBL2163449 | US9708370, CP-2B(v))
Affinity DataIC50:  6.66E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395014(CHEMBL2163454 | US9708370, 60 CP-3(iv))
Affinity DataIC50:  7.58E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395015(CHEMBL2163453 | US9708370, CP-2B(i))
Affinity DataIC50:  7.59E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394983(CHEMBL2163466)
Affinity DataIC50:  7.97E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395015(CHEMBL2163453 | US9708370, CP-2B(i))
Affinity DataIC50:  8.17E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395007(CHEMBL2163472)
Affinity DataIC50:  8.53E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394982(CHEMBL2163467)
Affinity DataIC50:  9.01E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395016(CHEMBL2163452 | US9708370, CP-2B(ii))
Affinity DataIC50:  9.48E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)
Affinity DataIC50:  9.61E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394989(CHEMBL2163460 | US9708370, 62 CP-AP-4)
Affinity DataIC50:  9.81E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394980(CHEMBL2163469)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394987(CHEMBL2163462 | US9708370, CP-AP-2)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394988(CHEMBL2163461 | US9708370, CP-AP-3)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394989(CHEMBL2163460 | US9708370, 62 CP-AP-4)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394990(CHEMBL2163459)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394991(CHEMBL2163438 | US9708370, 40 CP-1A(ii))
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394992(CHEMBL2163437)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50394998(CHEMBL2163481 | US9708370, DBG-253-5)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395000(CHEMBL2163479 | US9708370, DBG-253-2)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet glycoprotein 4(Rat)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395006(CHEMBL2163473)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395011(CHEMBL2163457 | US9708370, 57 CP-3(i))
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50395012(CHEMBL2163456 | US9708370, 58 CP-3(ii))
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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