Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50039978
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387167BDBM50387167(CHEMBL2047981)
Affinity DataIC50: 10.6nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387168BDBM50387168(CHEMBL2047982)
Affinity DataIC50: 13.1nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387178BDBM50387178(CHEMBL2047994)
Affinity DataIC50: 16.5nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387176BDBM50387176(CHEMBL2047992)
Affinity DataIC50: 22.1nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16673BDBM16673(BAY439006 | CHEMBL1336 | BAY 43-9006 | 4-[4-({[4-c...)
Affinity DataIC50: 24.3nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387175BDBM50387175(CHEMBL2047991)
Affinity DataIC50: 35.9nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387177BDBM50387177(CHEMBL2047993)
Affinity DataIC50: 46.7nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387164BDBM50387164(CHEMBL2047995)
Affinity DataIC50: 64.8nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387169BDBM50387169(CHEMBL2047983)
Affinity DataIC50: 69.2nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387166BDBM50387166(CHEMBL2047980)
Affinity DataIC50: 75.9nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387174BDBM50387174(CHEMBL2047990)
Affinity DataIC50: 77.7nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387170BDBM50387170(CHEMBL2047984)
Affinity DataIC50: 81.5nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387165BDBM50387165(CHEMBL2047979)
Affinity DataIC50: 87.8nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387171BDBM50387171(CHEMBL2047985)
Affinity DataIC50: 94.9nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387172BDBM50387172(CHEMBL2047986)
Affinity DataIC50: 120nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Academy of Military Medical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50387173BDBM50387173(CHEMBL2047988)
Affinity DataIC50: 148nMAssay Description:Inhibition of C-Raf kinase-mediated phosphorylation of Mek using [33P]gammaATP after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed