Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50040508
TargetHistone acetyltransferase p300(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50395259BDBM50395259(CHEMBL2163601)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50395258BDBM50395258(CHEMBL2163602)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50395261BDBM50395261(CHEMBL2163594)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Emory University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50395260BDBM50395260(CHEMBL2163598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed