Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50042803
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50384576(CHEMBL2036808)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431281(CHEMBL2347987)
Affinity DataIC50:  27nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation expressed in mouse NIH/3T3 cells after 2 hrs by immunoprecipitation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50384576(CHEMBL2036808)
Affinity DataIC50:  37nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50384576(CHEMBL2036808)
Affinity DataIC50:  48nMAssay Description:Inhibition of TYRO3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | 2-(2-hydroxyethyla...)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of MER (588 to 855) (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)
Affinity DataKd:  440nMAssay Description:Binding affinity to MET (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431278(CHEMBL2348264)
Affinity DataKd:  260nMAssay Description:Binding affinity to MER (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431279(CHEMBL2346680)
Affinity DataKd:  42nMAssay Description:Binding affinity to MER (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)
Affinity DataKd:  190nMAssay Description:Binding affinity to MER (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431278(CHEMBL2348264)
Affinity DataKd:  170nMAssay Description:Binding affinity to AXL (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431279(CHEMBL2346680)
Affinity DataKd:  39nMAssay Description:Binding affinity to AXL (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)
Affinity DataKd:  210nMAssay Description:Binding affinity to AXL (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431279(CHEMBL2346680)
Affinity DataKd:  4.00E+4nMAssay Description:Binding affinity to phosphorylated ABL1 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to phosphorylated ABL1 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431279(CHEMBL2346680)
Affinity DataKd:  6.60E+3nMAssay Description:Binding affinity to nonphosphorylated ABL1 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)
Affinity DataKd:  320nMAssay Description:Binding affinity to nonphosphorylated ABL1 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataKd:  93nMAssay Description:Binding affinity to TYRO3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to MER (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431279(CHEMBL2346680)
Affinity DataKd:  65nMAssay Description:Binding affinity to MET (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431278(CHEMBL2348264)
Affinity DataKd:  150nMAssay Description:Binding affinity to MET (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)
Affinity DataKd:  900nMAssay Description:Binding affinity to TYRO3 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataKd:  250nMAssay Description:Binding affinity to AXL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431278(CHEMBL2348264)
Affinity DataKd:  2.90E+3nMAssay Description:Binding affinity to TYRO3 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50431279(CHEMBL2346680)
Affinity DataKd:  200nMAssay Description:Binding affinity to TYRO3 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed