Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50040255
TargetMelanin-concentrating hormone receptor 1(RAT)
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50391543(CHEMBL2147477)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity at rat MCH1 receptor expressed in HEK 293T cells assessed as inhibition of MCH-induced Ca2+ mobilization after 10 mins by FLIPR a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50391542(CHEMBL2147476)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-MCH from human MCHR1 receptor expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed