Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50040314
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 24567BDBM24567(Tetrahydrolipstatin | CHEMBL175247 | Xenical | (2S...)
Affinity DataIC50: 220nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392476BDBM50392476(CHEMBL2152046)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392475BDBM50392475(CHEMBL2152045)
Affinity DataIC50: 2.46E+5nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392474BDBM50392474(CHEMBL2152044)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392477BDBM50392477(CHEMBL2152047)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085536BDBM50085536(Gallic Acid, F | 3,4,5-Trihydroxybenzoate, X | CHE...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Hokkaido University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4375BDBM4375(3,4-Dihydroxycinnamate, XVII | cid_689043 | Caffei...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of porcine pancreatic lipase using micellar solution of triolein as substrate preincubated for 5 mins before substrate addition measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed