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Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50040448
TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394369(CHEMBL2159781)
Affinity DataKi:  75.7nMAssay Description:Irreversible inhibition of human MAGL using p-nitrophenylpropionate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394369(CHEMBL2159781)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394387(CHEMBL2159800)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394382(CHEMBL2159805)
Affinity DataIC50:  2nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394370(CHEMBL2159780)
Affinity DataIC50:  3nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394367(CHEMBL2159783)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394387(CHEMBL2159800)
Affinity DataIC50:  3nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394394(CHEMBL2159776)
Affinity DataIC50:  4nMAssay Description:Inhibition of MAGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394375(CHEMBL2159812)
Affinity DataIC50:  7nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394389(CHEMBL2159798)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394381(CHEMBL2159806)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394373(CHEMBL2159777)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394371(CHEMBL2159779)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394382(CHEMBL2159805)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394384(CHEMBL2159803)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  10nMAssay Description:Inhibition of MAGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394386(CHEMBL2159801)
Affinity DataIC50:  10nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394385(CHEMBL2159802)
Affinity DataIC50:  11nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394390(CHEMBL2159797)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394371(CHEMBL2159779)
Affinity DataIC50:  12nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394383(CHEMBL2159804)
Affinity DataIC50:  12nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394376(CHEMBL2159811)
Affinity DataIC50:  13nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394368(CHEMBL2159782)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394370(CHEMBL2159780)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394386(CHEMBL2159801)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394363(CHEMBL2159787)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394385(CHEMBL2159802)
Affinity DataIC50:  17nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394374(CHEMBL2159813)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394357(CHEMBL2159795)
Affinity DataIC50:  19nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394366(CHEMBL2159784)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394389(CHEMBL2159798)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394362(CHEMBL2159788)
Affinity DataIC50:  20nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394390(CHEMBL2159797)
Affinity DataIC50:  21nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394384(CHEMBL2159803)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394373(CHEMBL2159777)
Affinity DataIC50:  23nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394388(CHEMBL2159799)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394368(CHEMBL2159782)
Affinity DataIC50:  30nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394372(CHEMBL2159778)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394363(CHEMBL2159787)
Affinity DataIC50:  32nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394372(CHEMBL2159778)
Affinity DataIC50:  33nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394388(CHEMBL2159799)
Affinity DataIC50:  33nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394362(CHEMBL2159788)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394375(CHEMBL2159812)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394378(CHEMBL2159809)
Affinity DataIC50:  36nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394360(CHEMBL2159790)
Affinity DataIC50:  38nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMonoglyceride lipase(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394358(CHEMBL2159794)
Affinity DataIC50:  41nMAssay Description:Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394381(CHEMBL2159806)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394376(CHEMBL2159811)
Affinity DataIC50:  44nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFatty-acid amide hydrolase 1(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50394378(CHEMBL2159809)
Affinity DataIC50:  58nMAssay Description:Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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