TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 3.77E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha ligand binding domain assessed as inhibition of CDCA-induced biotinylated SRC1 binding after 30 mins by HT...More data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 8.23E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha ligand binding domain assessed as inhibition of CDCA-induced biotinylated SRC1 binding after 30 mins by HT...More data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 1.29E+4nMAssay Description:Agonist activity at GST-tagged FXRalpha ligand binding domain assessed as biotinylated SRC1 binding after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 358nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 94nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 377nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 343nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
East China University Of Science And Technology
Curated by ChEMBL
East China University Of Science And Technology
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Agonist activity at FXRalpha expressed in HEK293 cells assessed as increase in transcriptional activity after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair