Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50040457
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394470(CHEMBL2160099)
Affinity DataIC50:  0.870nMAssay Description:Antagonist activity at CCR3 receptor in human eosinophils assessed as inhibition of CCL11-induced degranulation after 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394470(CHEMBL2160099)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394487(CHEMBL2160111)
Affinity DataIC50:  2.40nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394482(CHEMBL2159867)
Affinity DataIC50:  9.90nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394481(CHEMBL2159868)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394486(CHEMBL2159863)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394479(CHEMBL2160097)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394480(CHEMBL2159869)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394488(CHEMBL2160110)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394477(CHEMBL2160100)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394485(CHEMBL2159864)
Affinity DataIC50:  41nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394472(CHEMBL2160105)
Affinity DataIC50:  44nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394471(CHEMBL2160106)
Affinity DataIC50:  44nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394483(CHEMBL2159866)
Affinity DataIC50:  44nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394484(CHEMBL2159865)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394474(CHEMBL2160103)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394478(CHEMBL2160098)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394476(CHEMBL2160101)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394475(CHEMBL2160102)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394473(CHEMBL2160104)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394489(CHEMBL2160109)
Affinity DataIC50:  380nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394491(CHEMBL2160107)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50394490(CHEMBL2160108)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at CCR3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed