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Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50040240
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

LigandPNGBDBM50391185(CHEMBL2088663)
Affinity DataIC50:  91nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  150nMAssay Description:Inhibition of PI3K p110gamma by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

LigandPNGBDBM50391185(CHEMBL2088663)
Affinity DataIC50:  295nMAssay Description:Inhibition of PI3K p110gamma by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391186(CHEMBL2088664)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391187(CHEMBL2088665)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391195(CHEMBL2088673)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391184(CHEMBL2088662)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391187(CHEMBL2088665)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of PI3K p110gamma by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391194(CHEMBL2088672)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391196(CHEMBL2088674)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391197(CHEMBL2088675)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391200(CHEMBL2088661)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of PI3K p110gamma by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391192(CHEMBL2088670)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391191(CHEMBL2088669)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391182(CHEMBL2088659)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391200(CHEMBL2088661)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391186(CHEMBL2088664)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of PI3K p110gamma by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391181(CHEMBL2088658)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391183(CHEMBL2088660)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391199(CHEMBL2088677)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of PI3K p110alpha/p85alpha by fluorescence based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391186(CHEMBL2088664)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391187(CHEMBL2088665)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391188(CHEMBL2088666)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391189(CHEMBL2088667)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391190(CHEMBL2088668)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391191(CHEMBL2088669)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391192(CHEMBL2088670)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391193(CHEMBL2088671)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391194(CHEMBL2088672)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391195(CHEMBL2088673)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391196(CHEMBL2088674)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391197(CHEMBL2088675)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391198(CHEMBL2088676)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50391199(CHEMBL2088677)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A expressed in Escherichia coli using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391181(CHEMBL2088658)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391183(CHEMBL2088660)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391200(CHEMBL2088661)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391184(CHEMBL2088662)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391185(CHEMBL2088663)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391186(CHEMBL2088664)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391187(CHEMBL2088665)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391188(CHEMBL2088666)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391189(CHEMBL2088667)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391190(CHEMBL2088668)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391191(CHEMBL2088669)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391192(CHEMBL2088670)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391193(CHEMBL2088671)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50391194(CHEMBL2088672)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/P25 using myelin basic protein substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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