Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50040730
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399046BDBM50399046(CHEMBL2178862)
Affinity DataKi:  38nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399047BDBM50399047(CHEMBL2178856)
Affinity DataKi:  39nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399054BDBM50399054(CHEMBL2178851)
Affinity DataKi:  43nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399062BDBM50399062(CHEMBL2178843)
Affinity DataKi:  370nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399048BDBM50399048(CHEMBL2178861)
Affinity DataKi:  370nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399056BDBM50399056(CHEMBL2178849)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399051BDBM50399051(CHEMBL2178855)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399059BDBM50399059(CHEMBL2178846)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399049BDBM50399049(CHEMBL2178858)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399053BDBM50399053(CHEMBL2178852)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399060BDBM50399060(CHEMBL2178845)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Human)
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 92409BDBM92409(Epoxyazadiradione)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human MIFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399058BDBM50399058(CHEMBL2178847)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399065BDBM50399065(CHEMBL2178837)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399057BDBM50399057(CHEMBL2178848)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399050BDBM50399050(CHEMBL2178857)
Affinity DataKi:  7.70E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399072BDBM50399072(CHEMBL2178826)
Affinity DataKi:  8.60E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 92409BDBM92409(Epoxyazadiradione)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399055BDBM50399055(CHEMBL2178850)
Affinity DataKi:  1.13E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399071BDBM50399071(CHEMBL2178828)
Affinity DataKi:  1.55E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399069BDBM50399069(CHEMBL2178830)
Affinity DataKi:  1.93E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399074BDBM50399074(CHEMBL2178863)
Affinity DataKi:  2.06E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399066BDBM50399066(CHEMBL2178833)
Affinity DataKi:  2.29E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399073BDBM50399073(CHEMBL2178867)
Affinity DataKi:  2.54E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399070BDBM50399070(CHEMBL2178829)
Affinity DataKi:  2.86E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399067BDBM50399067(CHEMBL2178832)
Affinity DataKi:  4.34E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399063BDBM50399063(CHEMBL2178841)
Affinity DataKi:  5.72E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399064BDBM50399064(CHEMBL2178838)
Affinity DataKi:  6.76E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399052BDBM50399052(CHEMBL2178853)
Affinity DataKi:  9.33E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 61233BDBM61233(cid_367783 | SMR000496650 | MLS001164435 | 4-[(3,4...)
Affinity DataKi:  9.90E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Human)
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399047BDBM50399047(CHEMBL2178856)
Affinity DataKi:  1.01E+5nMAssay Description:Inhibition of human MIFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399061BDBM50399061(CHEMBL2178844)
Affinity DataKi:  1.22E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Plasmodium falciparum (isolate 3D7))
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399068BDBM50399068(CHEMBL2178831)
Affinity DataKi:  1.22E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum MIF expressed in Escherichia coli BL21 (DE3) assessed as ketonization of enol form of 4-HPP substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Human)
Yale University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399046BDBM50399046(CHEMBL2178862)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of human MIFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed