Compile Data Set for Download or QSAR
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Found 27 Enz. Inhib. hit(s) with all data for entry = 50040890
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity at progesterone receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401606(CHEMBL2203825)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401601(CHEMBL2203832)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401600(CHEMBL2203833)
Affinity DataIC50:  8nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401612(CHEMBL2203819)
Affinity DataIC50:  8nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at androgen receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401610(CHEMBL2203821)
Affinity DataIC50:  9nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401608(CHEMBL2203823)
Affinity DataIC50:  10nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401596(CHEMBL2203836)
Affinity DataIC50:  11.7nMAssay Description:Antagonist activity at progesterone receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401596(CHEMBL2203836)
Affinity DataIC50:  12nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401599(CHEMBL2203834)
Affinity DataIC50:  12nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401604(CHEMBL2203829)
Affinity DataIC50:  30nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401603(CHEMBL2203830)
Affinity DataIC50:  36nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401597(CHEMBL2203837)
Affinity DataIC50:  57nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401605(CHEMBL2203826)
Affinity DataIC50:  58nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401613(CHEMBL2203818)
Affinity DataIC50:  75nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401611(CHEMBL2203820)
Affinity DataIC50:  76nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401609(CHEMBL2203822)
Affinity DataIC50:  78nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401596(CHEMBL2203836)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at androgen receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at glucocorticoid receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401598(CHEMBL2203835)
Affinity DataIC50:  128nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401607(CHEMBL2203824)
Affinity DataIC50:  167nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at mineralocorticoid receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50375423(ASOPRISNIL)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at estrogen receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401602(CHEMBL2203831)
Affinity DataIC50: >3.00E+3nMAssay Description:Antagonist activity against progesterone receptor in human T47D cells by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401596(CHEMBL2203836)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at glucocorticoid receptor by cellular reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed