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Found 26 Enz. Inhib. hit(s) with all data for entry = 50040923
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402219(CHEMBL2204732)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402219(CHEMBL2204732)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402224(CHEMBL2204739)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402221(CHEMBL2204017)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402217(CHEMBL2204734)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402223(CHEMBL2204740)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402220(CHEMBL2204018)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402220(CHEMBL2204018)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402222(CHEMBL2204741)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402225(CHEMBL2204738)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402217(CHEMBL2204734)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402223(CHEMBL2204740)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402220(CHEMBL2204018)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402220(CHEMBL2204018)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402226(CHEMBL2204737)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402218(CHEMBL2204733)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402221(CHEMBL2204017)
Affinity DataIC50:  9nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402224(CHEMBL2204739)
Affinity DataIC50:  10nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402225(CHEMBL2204738)
Affinity DataIC50:  16nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402222(CHEMBL2204741)
Affinity DataIC50:  18nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402218(CHEMBL2204733)
Affinity DataIC50:  23nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402226(CHEMBL2204737)
Affinity DataIC50:  54nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402227(CHEMBL2204736)
Affinity DataIC50:  406nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402227(CHEMBL2204736)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402228(CHEMBL2204735)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(DABCYL)-Arg as substrate incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50402228(CHEMBL2204735)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 60 mins by competitive radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed