Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50042343
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424331(CHEMBL2314497)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50304501(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424324(CHEMBL2314761)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50304501(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424340(CHEMBL2314772)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424327(CHEMBL2314501)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424325(CHEMBL2314760)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424338(CHEMBL2314774)
Affinity DataKi:  2.64E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424341(CHEMBL2314771)
Affinity DataKi:  2.67E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424326(CHEMBL2314759)
Affinity DataKi:  2.93E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424337(CHEMBL2314775)
Affinity DataKi:  3.28E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424336(CHEMBL2314776)
Affinity DataKi:  3.32E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424335(CHEMBL2314777)
Affinity DataKi:  3.73E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424330(CHEMBL2314498)
Affinity DataKi:  4.07E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424339(CHEMBL2314773)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424323(CHEMBL2314762)
Affinity DataKi:  5.95E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424334(CHEMBL2314494)
Affinity DataKi:  7.32E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424320(CHEMBL2314765)
Affinity DataKi:  8.13E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424328(CHEMBL2314500)
Affinity DataKi:  8.72E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424333(CHEMBL2314495)
Affinity DataKi:  8.99E+3nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424322(CHEMBL2314763)
Affinity DataKi:  1.05E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424319(CHEMBL2314766)
Affinity DataKi:  2.52E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424332(CHEMBL2314496)
Affinity DataKi:  3.61E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424321(CHEMBL2314764)
Affinity DataKi:  3.64E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424318(CHEMBL2314767)
Affinity DataKi:  4.42E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424342(CHEMBL2314770)
Affinity DataKi:  4.59E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424329(CHEMBL2314499)
Affinity DataKi:  4.80E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424317(CHEMBL2314768)
Affinity DataKi:  6.79E+4nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424331(CHEMBL2314497)
Affinity DataKi:  8.47E+4nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50424316(CHEMBL2314769)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed