Compile Data Set for Download or QSAR
Report error Found 162 Enz. Inhib. hit(s) with all data for entry = 50042364
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 29nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 80nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424711BDBM50424711(CHEMBL2314163)
Affinity DataIC50: 410nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424676BDBM50424676(CHEMBL2313912)
Affinity DataIC50: 500nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424671BDBM50424671(CHEMBL2313917)
Affinity DataIC50: 610nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424660BDBM50424660(CHEMBL2313884)
Affinity DataIC50: 660nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424676BDBM50424676(CHEMBL2313912)
Affinity DataIC50: 680nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424663BDBM50424663(CHEMBL2313925)
Affinity DataIC50: 710nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424664BDBM50424664(CHEMBL2313924)
Affinity DataIC50: 710nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424660BDBM50424660(CHEMBL2313884)
Affinity DataIC50: 790nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 800nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424707BDBM50424707(CHEMBL2314167)
Affinity DataIC50: 880nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 900nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424665BDBM50424665(CHEMBL2313923)
Affinity DataIC50: 930nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424680BDBM50424680(CHEMBL2313908)
Affinity DataIC50: 930nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424711BDBM50424711(CHEMBL2314163)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424707BDBM50424707(CHEMBL2314167)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424665BDBM50424665(CHEMBL2313923)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424668BDBM50424668(CHEMBL2313920)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424670BDBM50424670(CHEMBL2313918)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424703BDBM50424703(CHEMBL2313885)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424664BDBM50424664(CHEMBL2313924)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424662BDBM50424662(CHEMBL2313926)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424680BDBM50424680(CHEMBL2313908)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424703BDBM50424703(CHEMBL2313885)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424671BDBM50424671(CHEMBL2313917)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424694BDBM50424694(CHEMBL2313894)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424697BDBM50424697(CHEMBL2313891)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424679BDBM50424679(CHEMBL2313909)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424697BDBM50424697(CHEMBL2313891)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424679BDBM50424679(CHEMBL2313909)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424670BDBM50424670(CHEMBL2313918)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424682BDBM50424682(CHEMBL2313906)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424662BDBM50424662(CHEMBL2313926)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424681BDBM50424681(CHEMBL2313907)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424669BDBM50424669(CHEMBL2313919)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424661BDBM50424661(CHEMBL2313927)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424666BDBM50424666(CHEMBL2313922)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424705BDBM50424705(CHEMBL2314169)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424706BDBM50424706(CHEMBL2314168)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424704BDBM50424704(CHEMBL2314170)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424709BDBM50424709(CHEMBL2314165)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424710BDBM50424710(CHEMBL2314164)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424708BDBM50424708(CHEMBL2314166)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant CLK1-GST expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424677BDBM50424677(CHEMBL2313911)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424678BDBM50424678(CHEMBL2313910)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424675BDBM50424675(CHEMBL2313913)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424667BDBM50424667(CHEMBL2313921)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Rouen Normandy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424673BDBM50424673(CHEMBL2313915)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A-GST expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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