Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50042388
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425232(CHEMBL2314836)
Affinity DataIC50:  9.80nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50:  74nMAssay Description:Binding affinity to Y1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50425231(CHEMBL2314835)
Affinity DataIC50:  80nMAssay Description:Displacement of [125I]-NPY from Y1 receptor in human MCF7 cells in presence of 1 uM BBNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed