Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50042502
TargetSerine/threonine-protein kinase PLK1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50426931(CHEMBL2323729 | US20230365568, Compound 6a)
Affinity DataIC50: 5.27E+3nMAssay Description:Inhibition of Plk1 polo-box domain in human HeLa cells/biotin-GGGGG-PLHSpT interaction incubated for 30 mins measured after 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.24E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged Plk1 in presence of 62.5 uM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged Plk1 in presence of 3.12 mM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50426930(CHEMBL2324036)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged Plk1 in presence of 3.12 mM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50426930(CHEMBL2324036)
Affinity DataIC50: 1.46E+5nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged Plk1 in presence of 62.5 uM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50426930(CHEMBL2324036)
Affinity DataIC50: 1.51E+5nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed