Compile Data Set for Download or QSAR
maximum 50k data
Found 175 Enz. Inhib. hit(s) with all data for entry = 50042448
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  5nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426336(CHEMBL2321952)
Affinity DataIC50:  70nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426339(CHEMBL2321961)
Affinity DataIC50:  100nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426339(CHEMBL2321961)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426337(CHEMBL1233659)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

LigandPNGBDBM50426338(CHEMBL2321958)
Affinity DataIC50:  130nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426338(CHEMBL2321958)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426334(CHEMBL2321948)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426334(CHEMBL2321948)
Affinity DataIC50:  200nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426337(CHEMBL1233659)
Affinity DataIC50:  210nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426338(CHEMBL2321958)
Affinity DataIC50:  220nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426312(CHEMBL2321951)
Affinity DataIC50:  300nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426336(CHEMBL2321952)
Affinity DataIC50:  310nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426336(CHEMBL2321952)
Affinity DataIC50:  350nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426332(CHEMBL2321964)
Affinity DataIC50:  400nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426332(CHEMBL2321964)
Affinity DataIC50:  400nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426312(CHEMBL2321951)
Affinity DataIC50:  400nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426335(CHEMBL2321878)
Affinity DataIC50:  410nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426336(CHEMBL2321952)
Affinity DataIC50:  420nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426312(CHEMBL2321951)
Affinity DataIC50:  520nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426336(CHEMBL2321952)
Affinity DataIC50:  530nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426310(CHEMBL2321967)
Affinity DataIC50:  580nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426331(CHEMBL2321965)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426315(CHEMBL2321962)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426331(CHEMBL2321965)
Affinity DataIC50:  600nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426313(CHEMBL2321959)
Affinity DataIC50:  630nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426313(CHEMBL2321959)
Affinity DataIC50:  800nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426334(CHEMBL2321948)
Affinity DataIC50:  800nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426312(CHEMBL2321951)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426330(CHEMBL2321974)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426314(CHEMBL2321968)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426334(CHEMBL2321948)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426335(CHEMBL2321878)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426333(CHEMBL2321945)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426333(CHEMBL2321945)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50191405((2'Z,3'E)-7-bromoindirubin-3'-oxime | CHEMBL373834)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426314(CHEMBL2321968)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426332(CHEMBL2321964)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426335(CHEMBL2321878)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426315(CHEMBL2321962)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426339(CHEMBL2321961)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426330(CHEMBL2321974)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426314(CHEMBL2321968)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50426313(CHEMBL2321959)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human recombinant GST-fused DYRK2 expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50191405((2'Z,3'E)-7-bromoindirubin-3'-oxime | CHEMBL373834)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426314(CHEMBL2321968)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50426331(CHEMBL2321965)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrate after 30 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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