TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to mouse GAT1 expressed in HEK293 cells membranes using LC-ESI-MS/MS analysis by [2H10]NO711 binding inhibition assayMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mus musculus)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair