Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50005288
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490702BDBM50490702(CHEMBL2337686)
Affinity DataIC50: 0.347nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490707BDBM50490707(BDBM50490709 | CHEMBL2337687)
Affinity DataIC50: 0.912nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490707BDBM50490707(BDBM50490709 | CHEMBL2337687)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490706BDBM50490706(CHEMBL2337677)
Affinity DataIC50: 4.30nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82258BDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 5.60nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490699BDBM50490699(CHEMBL2337681)
Affinity DataIC50: 43nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490704BDBM50490704(CHEMBL2337684)
Affinity DataIC50: 331nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490698BDBM50490698(CHEMBL2337683)
Affinity DataIC50: 417nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490708BDBM50490708(CHEMBL2337685)
Affinity DataIC50: 501nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490701BDBM50490701(CHEMBL2337679)
Affinity DataIC50: 708nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490703BDBM50490703(CHEMBL2337678)
Affinity DataIC50: 832nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490705BDBM50490705(CHEMBL2337682)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
University of Patras

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50490700BDBM50490700(CHEMBL2337680)
Affinity DataIC50: 6.46E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]-ANG2 from human Angiotensin 2 type-1 receptor expressed in HEK293 cells after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed