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Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50042538
TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427452(CHEMBL2326941)
Affinity DataIC50:  4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM53163((3E)-5-bromo-1H-indole-2,3-dione 3-[(3-methylpheny...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human full length PDE4B expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427451(CHEMBL2326942)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427450(CHEMBL2326943)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM53163((3E)-5-bromo-1H-indole-2,3-dione 3-[(3-methylpheny...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427450(CHEMBL2326943)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human full length PDE4B expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427448(CHEMBL2326945)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human full length PDE4B expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427449(CHEMBL2326944)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human full length PDE4B expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427451(CHEMBL2326942)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human full length PDE4B expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427449(CHEMBL2326944)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427448(CHEMBL2326945)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427447(CHEMBL2326946)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of human full length PDE4B expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPhosphodiesterase(Trypanosoma brucei)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50427447(CHEMBL2326946)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of Trypanosoma brucei full length PDEB1 expressed in insect SF21 cells using cAMP as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed