Compile Data Set for Download or QSAR
maximum 50k data
Found 61 Enz. Inhib. hit(s) with all data for entry = 50042846
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432133(CHEMBL2349589)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432132(CHEMBL2349590)
Affinity DataEC50:  130nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432135(CHEMBL2349587)
Affinity DataEC50:  550nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432136(CHEMBL2349586)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432137(CHEMBL2349585)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432138(CHEMBL2349584)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432139(CHEMBL2349583)
Affinity DataEC50:  300nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432140(CHEMBL2349582)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432141(CHEMBL2349581)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432142(CHEMBL2349580)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432143(CHEMBL2349579)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432144(CHEMBL2349578)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432145(CHEMBL2349577)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432146(CHEMBL2346788)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432147(CHEMBL2346787)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432148(CHEMBL2346786)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432149(CHEMBL2346785)
Affinity DataEC50:  1.00E+4nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432150(CHEMBL2346784)
Affinity DataEC50:  800nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432151(CHEMBL2346783)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432152(CHEMBL2346782)
Affinity DataEC50:  1.50E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432153(CHEMBL2346781)
Affinity DataEC50:  1.00E+4nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432154(CHEMBL2346780)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432155(CHEMBL2346779)
Affinity DataEC50:  1.50E+4nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432156(CHEMBL2346666)
Affinity DataEC50:  6.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432157(CHEMBL2346778)
Affinity DataEC50:  2.00E+4nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432158(CHEMBL2346777)
Affinity DataEC50:  3.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432159(CHEMBL2346776)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432160(CHEMBL2346775)
Affinity DataEC50:  1.50E+4nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432161(CHEMBL2346774)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432162(1-(3,3-diphenylpropyl)-3-p-tolylurea | CHEMBL23467...)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432163(CHEMBL2346772)
Affinity DataEC50:  3.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432164(CHEMBL2346771)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432165(CHEMBL2346770)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432166(CHEMBL2346769)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432167(CHEMBL2346768)
Affinity DataEC50:  6.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432168(CHEMBL2346767)
Affinity DataEC50:  1.50E+4nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432169(CHEMBL2346766)
Affinity DataEC50:  8.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50416875(AMG-073 | AMG073 HCL | CINACALCET | CINACALCET HYD...)
Affinity DataEC50:  80nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM61401(3,3-diphenyl-N-(1-phenylethyl)-1-propanamine;hydro...)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50299670((R)-3-(2-chlorophenyl)-N-(1-(3-methoxyphenyl)ethyl...)
Affinity DataEC50:  80nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432112(CHEMBL2349576)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432113(CHEMBL2349575)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432114(CHEMBL2349574)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432115(CHEMBL2349573)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432116(CHEMBL2346765)
Affinity DataEC50:  600nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432117(CHEMBL2349605)
Affinity DataEC50:  300nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432118(CHEMBL2349604)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432119(CHEMBL2349603)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432120(CHEMBL2349602)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432121(CHEMBL2349601)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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