Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with all data for entry = 50042777
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Heptares Therapeutics

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKd:  5.60E+3nMAssay Description:Binding affinity to His-tagged human beta1 adrenergic receptor expressed in HEK293 cell membranes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Heptares Therapeutics

Curated by ChEMBL
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKd:  1.60E+4nMAssay Description:Binding affinity to His-tagged human beta1 adrenergic receptor expressed in HEK293 cell membranes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed