Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50042777
TargetBeta-1 adrenergic receptor(Human)
Heptares Therapeutics

Curated by ChEMBL
LigandPNGBDBM50014407(2-Piperazin-1-yl-quinoline (Quipazine) | CHEMBL187...)
Affinity DataKd:  5.60E+3nMAssay Description:Binding affinity to His-tagged human beta1 adrenergic receptor expressed in HEK293 cell membranes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Heptares Therapeutics

Curated by ChEMBL
LigandPNGBDBM50035057(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazine |...)
Affinity DataKd:  1.60E+4nMAssay Description:Binding affinity to His-tagged human beta1 adrenergic receptor expressed in HEK293 cell membranes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed