Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50042781
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430945(CHEMBL2336987)
Affinity DataIC50:  460nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430946(CHEMBL2336980)
Affinity DataIC50:  990nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430944(CHEMBL2336966)
Affinity DataIC50:  1.46E+3nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430944(CHEMBL2336966)
Affinity DataIC50:  4.45E+3nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430946(CHEMBL2336980)
Affinity DataIC50:  2.56E+4nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430945(CHEMBL2336987)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed